Pre-arrayed esiRNA sub-libraries

Our pre-arrayed human and mouse sub-libraries provide state-of-the-art silencing triggers to study the function of an entire protein family, or biological process, such as epigenetics, ubiquitin conjugation, ion channels, membrane transporters, nuclear receptors, receptors in general, transcription factors,  transporters, proteases, kinases, and phosphatases. All of these sub-libraries are druggable.

Exemplary human druggable sub-libraries with their targets are listed below. For other, or custom sub-libraries please inquire.

esiRNA IDGene NameGene DescriptionEnsembl ID
HU-02595-1ARandrogen receptorENSG00000169083
HU-14165-1ESR1estrogen receptor 1ENSG00000091831
HU-90008-1ESR2Estrogen receptor 2 (ER beta)ENSG00000140009
HU-10728-1ESRRAestrogen-related receptor alphaENSG00000173153
HU-04474-1ESRRBestrogen-related receptor betaENSG00000119715
HU-90009-1ESRRGEstrogen-related receptor gammaENSG00000196482
HU-06674-1HNF4Ahepatocyte nuclear factor 4, alphaENSG00000101076
HU-09225-1HNF4Ghepatocyte nuclear factor 4, gammaENSG00000164749
HU-12211-1NR0B1nuclear receptor subfamily 0, group B, member 1ENSG00000169297
HU-15663-1NR0B2nuclear receptor subfamily 0, group B, member 2ENSG00000131910
HU-14341-1NR1D1nuclear receptor subfamily 1, group D, member 1ENSG00000126368
HU-04844-1NR1D2nuclear receptor subfamily 1, group D, member 2ENSG00000174738
HU-01834-1NR1H2nuclear receptor subfamily 1, group H, member 2ENSG00000131408
HU-13463-1NR1H3nuclear receptor subfamily 1, group H, member 3ENSG00000025434
HU-13316-1NR1H4nuclear receptor subfamily 1, group H, member 4ENSG00000012504
HU-08147-1NR1I2nuclear receptor subfamily 1, group I, member 2ENSG00000144852
HU-13906-1NR1I3nuclear receptor subfamily 1, group I, member 3ENSG00000143257
HU-08565-1NR2C1nuclear receptor subfamily 2, group C, member 1ENSG00000120798
HU-04202-1NR2C2nuclear receptor subfamily 2, group C, member 2ENSG00000177463
HU-13025-1NR2E1nuclear receptor subfamily 2, group E, member 1ENSG00000112333
HU-13277-1NR2E3nuclear receptor subfamily 2, group E, member 3ENSG00000031544
HU-90006-1NR2F1nuclear receptor subfamily 2, group F, member 1ENSG00000175745
HU-02364-1NR2F2nuclear receptor subfamily 2, group F, member 2ENSG00000185551
HU-90007-1NR2F6Nuclear receptor subfamily 2, group F, member 6ENSG00000160113
HU-06800-1NR3C1nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor)ENSG00000113580
HU-08859-1NR3C2nuclear receptor subfamily 3, group C, member 2ENSG00000151623
HU-15723-1NR4A1nuclear receptor subfamily 4, group A, member 1ENSG00000123358
HU-00873-1NR4A2nuclear receptor subfamily 4, group A, member 2ENSG00000153234
HU-90011-1NR4A3Nuclear receptor subfamily 4, group A, member 3ENSG00000119508
HU-14253-1NR5A1nuclear receptor subfamily 5, group A, member 1ENSG00000136931
HU-06607-1NR5A2nuclear receptor subfamily 5, group A, member 2ENSG00000116833
HU-05095-1NR6A1nuclear receptor subfamily 6, group A, member 1ENSG00000148200
HU-90010-1PGRProgesterone receptorENSG00000082175
HU-15182-1PPARAperoxisome proliferator-activated receptor alphaENSG00000186951
HU-05879-1PPARDperoxisome proliferator-activated receptor deltaENSG00000112033
HU-09771-1PPARGperoxisome proliferator-activated receptor gammaENSG00000132170
HU-06427-1RARAretinoic acid receptor, alphaENSG00000131759
HU-06658-1RARBretinoic acid receptor, betaENSG00000077092
HU-15819-1RARGretinoic acid receptor, gammaENSG00000172819
HU-07274-1RORARAR-related orphan receptor AENSG00000069667
HU-10108-1RORBRAR-related orphan receptor BENSG00000198963
HU-09384-1RORCRAR-related orphan receptor CENSG00000143365
HU-15326-1RXRAretinoid X receptor, alphaENSG00000186350
HU-21995-1RXRBretinoid X receptor, betaENSG00000204231
HU-06498-1RXRGretinoid X receptor, gammaENSG00000143171
HU-01376-1THRAthyroid hormone receptor, alphaENSG00000126351
HU-08346-1THRBthyroid hormone receptor, betaENSG00000151090
HU-01044-1VDRvitamin D (1,25- dihydroxyvitamin D3) receptorENSG00000111424